ETHAN S. BURSTEIN: search on Z-Library

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1

Bromazepam pharmacokinetics: Influence of age, gender, oral contraceptives, cimetidine, and propranolol

Ochs, Hermann R, Greenblatt, David J, Friedman, H, Burstein, Ethan S, Locniskar, Ann, Harmatz, Jerold S, Shader, Richard I

Journal:

Clinical Pharmacology & Therapeutics

Year:

1987

Language:

english

File:

PDF, 698 KB

english, 1987

2

Pharmacokinetics and CSF Entry of Flurazepam in Dogs

Ochs, Hermann R., Greenblatt, David J., Burstein, Ethan S., Eichelkraut, Wolfgang, Hahn, Norbert

Journal:

Year:

1988

Language:

english

File:

PDF, 776 KB

english, 1988

3

Pimavanserin, a 5HT 2A receptor inverse agonist, rapidly suppresses AÎ² production and related pathology in a mouse model of Alzheimerâs disease

Yuede, Carla M., Wallace, Clare E., Davis, Todd A., Gardiner, Woodrow D., Hettinger, Jane C., Edwards, Hannah M., Hendrix, Rachel D., Doherty, Brookelyn M., Yuede, Kayla M., Burstein, Ethan S., Cirrit

Journal:

Journal of Neurochemistry

Year:

2020

File:

PDF, 24.25 MB

2020

4

Bexarotene prodrugs: Targeting through cleavage by NQO1 (DT-diaphorase)

Schäfer, Anja, Burstein, Ethan S., Olsson, Roger

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2014

Language:

english

File:

PDF, 897 KB

english, 2014

5

Discovery of potential antipsychotic agents possessing pro-cognitive properties

Jelveh Lameh, Krista McFarland, Jorgen Ohlsson, Fredrik Ek, Fabrice Piu, Ethan S. Burstein, Ali Tabatabaei, Roger Olsson, Stefania Risso Bradley, Douglas W. Bonhaus

Journal:

Naunyn-Schmiedeberg's Archives of Pharmacology

Year:

2012

Language:

english

File:

PDF, 352 KB

english, 2012

6

Characterization of the Mas-related gene family: structural and functional conservation of human and rhesus MrgX receptors

Ethan S Burstein, Thomas R Ott, Michele Feddock, Jian-Nong Ma, Steve Fuhs, Steven Wong, Hans H Schiffer, Mark R Brann, Norman R Nash

Journal:

British Journal of Pharmacology

Year:

2006

Language:

english

File:

PDF, 232 KB

english, 2006

7

Chiral Dihydrobenzofuran Acids Show Potent Retinoid X Receptor–Nuclear Receptor Related 1 Protein Dimer Activation

Sundén, Henrik, Schäfer, Anja, Scheepstra, Marcel, Leysen, Seppe, Malo, Marcus, Ma, Jian-Nong, Burstein, Ethan S., Ottmann, Christian, Brunsveld, Luc, Olsson, Roger

Journal:

Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 2.17 MB

english, 2016

8

Chemical genomics: massively parallel technologies for rapid lead identification and target validation

Uli Hacksell, Norman Nash, Ethan S. Burstein, Fabrice Piu, Glenn Croston, Mark R. Brann

Journal:

Year:

2002

Language:

english

File:

PDF, 544 KB

english, 2002

9

Reversal of morphine tolerance by a compound with NPFF receptor subtype-selective actions

Malin, David H., Henceroth, Mallori M., Izygon, Jonathan J., Nghiem, Duyen M., Moon, Will D., Anderson, Andrea P., Madison, Caitlin A., Goyarzu, Pilar, Ma, Jian-Nong, Burstein, Ethan S.

Journal:

Neuroscience Letters

Year:

2015

Language:

english

File:

PDF, 450 KB

english, 2015

10

Optimization of isochromanone based urotensin II receptor agonists

Fredrik Lehmann, Erika A. Currier, Roger Olsson, Jian-Nong Ma, Ethan S. Burstein, Uli Hacksell, Kristina Luthman

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 557 KB

english, 2010

11

Structure/Function Relationships of a G-Protein Coupling Pocket Formed by the Third Intracellular Loop of the m5 Muscarinic Receptor †

Burstein, Ethan S., Spalding, Tracy A., Brann, Mark R.

Journal:

Year:

1998

Language:

english

File:

PDF, 76 KB

english, 1998

12

A subtype-specific Neuropeptide FF receptor antagonist attenuates morphine and nicotine withdrawal syndrome in the rat

Malin, David H., Henceroth, Mallori M., Elayoubi, Joanne, Campbell, Joseph R., Anderson, Andrea, Goyarzu, Pilar, Izygon, Jonathon, Madison, Caitlin A., Ward, Christopher P., Burstein, Ethan S.

Journal:

Neuroscience Letters

Year:

2018

Language:

english

File:

PDF, 431 KB

english, 2018

13

Low Dose Bexarotene Treatment Rescues Dopamine Neurons and Restores Behavioral Function in Models of Parkinson’s Disease

McFarland, Krista, Spalding, Tracy A., Hubbard, David, Ma, Jian-Nong, Olsson, Roger, Burstein, Ethan S.

Journal:

ACS Chemical Neuroscience

Year:

2013

Language:

english

File:

PDF, 1.46 MB

english, 2013

14

Discovery of novel peptide/receptor interactions: identification of PHM-27 as a potent agonist of the human calcitonin receptor

Jian-Nong Ma, Erika A Currier, Anthony Essex, Michele Feddock, Tracy A Spalding, Norman R Nash, Mark R Brann, Ethan S Burstein

Journal:

Biochemical Pharmacology

Year:

2004

Language:

english

File:

PDF, 142 KB

english, 2004

15

The human angiotensin AT1 receptor supports G protein-independent extracellular signal-regulated kinase 1/2 activation and cellular proliferation

Jakob Lerche Hansen, Mark Aplin, Jonas Tind Hansen, Gitte Lund Christensen, Marie Mi Bonde, Mikael Schneider, Stig Haunsø, Hans H. Schiffer, Ethan S. Burstein, David M. Weiner, Søren P. Sheikh

Journal:

European Journal of Pharmacology

Year:

2008

Language:

english

File:

PDF, 856 KB

english, 2008

16

On the Discovery and Development of Pimavanserin: A Novel Drug Candidate for Parkinson’s Psychosis

Hacksell, Uli, Burstein, Ethan S., McFarland, Krista, Mills, Roger G., Williams, Hilde

Journal:

Neurochemical Research

Year:

2014

Language:

english

File:

PDF, 1.01 MB

english, 2014

17

Discovery of Potent and Selective Small-Molecule PAR-2 Agonists

Seitzberg, Jimmi Gerner, Knapp, Anne Eeg, Lund, Birgitte Winther, Mandrup Bertozzi, Sine, Currier, Erika A., Ma, Jian-Nong, Sherbukhin, Vladimir, Burstein, Ethan S., Olsson, Roger

Journal:

Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 171 KB

english, 2008

18

Constitutive Activity of Muscarinic Acetylcholine Receptors

Spalding, Tracy A., Burstein, Ethan S.

Journal:

Journal of Receptor and Signal Transduction Research

Year:

2006

Language:

english

File:

PDF, 580 KB

english, 2006

19

Preclinical PET Neuroimaging of [ 11 C]Bexarotene

Rotstein, Benjamin H., Placzek, Michael S., Krishnan, Hema S., Pekošak, Aleksandra, Collier, Thomas Lee, Wang, Changning, Liang, Steven H., Burstein, Ethan S., Hooker, Jacob M., Vasdev, Neil

Journal:

Molecular Imaging

Year:

2016

Language:

english

File:

PDF, 345 KB

english, 2016

20

Prostaglandins and cannabis—XI Inhibition of Δ1-tetrahydrocannabinol-induced hypotension by aspirin

Sumner Burstein, Kent Ozman, Ethan Burstein, Nancy Palermo, Emil Smith

Journal:

Biochemical Pharmacology

Year:

1982

Language:

english

File:

PDF, 188 KB

english, 1982

21

AC-186, a Selective Nonsteroidal Estrogen Receptor β Agonist, Shows Gender Specific Neuroprotection in a Parkinson’s Disease Rat Model

McFarland, Krista, Price, Diana L., Davis, Christopher N., Ma, Jian-Nong, Bonhaus, Douglas W., Burstein, Ethan S., Olsson, Roger

Journal:

ACS Chemical Neuroscience

Year:

2013

Language:

english

File:

PDF, 2.03 MB

english, 2013

22

Design of a Highly Selective and Potent Class of Non-planar Estrogen Receptor β Agonists

Sundén, Henrik, Ma, Jian-Nong, Hansen, Lars K., Gustavsson, Anna-Lena, Burstein, Ethan S., Olsson, Roger

Journal:

Year:

2013

Language:

english

File:

PDF, 1.01 MB

english, 2013

23

Inverse agonists of the 5-HT2A receptor reduce nicotine withdrawal signs in rats

Malin, David, Henceroth, Mallori, Rao, Gadam Srinivas, Campbell, Joseph, Ma, Jian-Nong, Tsai, Ping-Hsun, Kishbaugh, Jordan C., Burstein, Ethan S.

Journal:

Neuroscience Letters

Year:

2019

Language:

english

File:

PDF, 1.35 MB

english, 2019

24

Pharmacology of N-desmethylclozapine

Jelveh Lameh, Ethan S. Burstein, Eve Taylor, David M. Weiner, Kimberly E. Vanover, Douglas W. Bonhaus

Journal:

Pharmacology & Therapeutics

Year:

2007

Language:

english

File:

PDF, 217 KB

english, 2007

25

Integrative Functional Assays, Chemical Genomics and High Throughput Screening: Harnessing Signal Transduction Pathways to a Common HTS Readout

Burstein, Ethan, Piu, Fabrice, Ma, Jian-Nong, Weissman, Jacques, Currier, Erika, Nash, Norman, Weiner, David, Spalding, Tracy, Schiffer, Hans, Del Tredici, Andria, Brann, Mark

Journal:

Current Pharmaceutical Design

Year:

2006

Language:

english

File:

PDF, 356 KB

english, 2006

26

Dronedarone Modulates M1 and M3 Muscarinic Receptors with Subtype Selectivity, Functional Selectivity, and Probe Dependence

Jayasuriya, Gihan M., Elmslie, Gwendolynne, Burstein, Ethan S., Ellis, John

Journal:

Year:

2017

Language:

english

File:

PDF, 200 KB

english, 2017

27

Simplified gas chromatographic analysis of ethanol in blood and tissue

Ethan S. Burstein, David J. Greenblatt

Journal:

Journal of Chromatography B: Biomedical Sciences and Applications

Year:

1989

Language:

english

File:

PDF, 272 KB

english, 1989

28

Constitutive activation of muscarinic receptors by the G-protein Gq

Ethan S. Burstein, Tracy A. Spalding, Hans Braüner-Osborne, Mark R. Brann

Journal:

Year:

1995

Language:

english

File:

PDF, 267 KB

english, 1995

29

Characterization of a Guanine Nucleotide-Releasing Factor and a GTPase- Activating Protein that are Specific for the Ras-Related Protein p25rab3A

Ethan S. Burstein and Ian G. Macara

Journal:

Proceedings of the National Academy of Sciences

Year:

1992

Language:

english

File:

PDF, 997 KB

english, 1992

30

Constitutive Activation of the m5 Muscarinic Receptor by a Series of Mutations at the Extracellular End of Transmembrane 6 †

Spalding, Tracy A., Burstein, Ethan S., Wells, James W., Brann, Mark R.

Journal:

Year:

1997

Language:

english

File:

PDF, 165 KB

english, 1997

31

Discovery of a class of calcium sensing receptor positive allosteric modulators; 1-(benzothiazol-2-yl)-1-phenylethanols

Magnus Gustafsson, Jacob Jensen, Sine M. Bertozzi, Erika A. Currier, Jian-Nong Ma, Ethan S. Burstein, Roger Olsson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 620 KB

english, 2010

32

Trazodone kinetics: Effect of age, gender, and obesity

Greenblatt, David J, Friedman, H, Burstein, Ethan S, Scavone, Joseph M, Blyden, Gershwin T, Ochs, Hermann R, Miller, Lawrence G, Harmatz, Jerold S, Shader, Richard I

Journal:

Clinical Pharmacology & Therapeutics

Year:

1987

Language:

english

File:

PDF, 512 KB

english, 1987

33

The ras-related GTPase rac1 regulates a proliferative pathway selectively utilized by G-protein coupled receptors

Burstein, Ethan S, Hesterberg, Diane J, Gutkind, J Silvio, Brann, Mark R, Currier, Erika A, Messier, Terri L

Journal:

Year:

1998

Language:

english

File:

PDF, 361 KB

english, 1998

34

ChemInform Abstract: Design of a Highly Selective and Potent Class of Non-planar Estrogen Receptor β Agonists.

Sunden, Henrik, Ma, Jian-Nong, Hansen, Lars K., Gustavsson, Anna-Lena, Burstein, Ethan S., Olsson, Roger

Journal:

Year:

2013

File:

PDF, 35 KB

2013

35

Identification of novel selective V2 receptor non-peptide agonists

Andria L. Del Tredici, Kim E. Vanover, Anne E. Knapp, Sine M. Bertozzi, Norman R. Nash, Ethan S. Burstein, Jelveh Lameh, Erika A. Currier, Robert E. Davis, Mark R. Brann, Nina Mohell, Roger Olsson, Fa

Journal:

Biochemical Pharmacology

Year:

2008

Language:

english

File:

PDF, 440 KB

english, 2008

36

II. In vitro evidence that (−)-OSU6162 and (+)-OSU6162 produce their behavioral effects through 5-HT2A serotonin and D2 dopamine receptors

Ethan S. Burstein, Maria L. Carlsson, Michelle Owens, Jian-Nong Ma, Hans H. Schiffer, Arvid Carlsson, Uli Hacksell

Journal:

Journal of Neural Transmission

Year:

2011

Language:

english

File:

PDF, 1.90 MB

english, 2011

37

An Angiotensin II type 1 receptor activation switch patch revealed through Evolutionary Trace analysis

Marie Mi Bonde, Rong Yao, Jian-Nong Ma, Srinivasan Madabushi, Stig Haunsø, Ethan S. Burstein, Jennifer L. Whistler, Søren P. Sheikh, Olivier Lichtarge, Jakob Lerche Hansen

Journal:

Biochemical Pharmacology

Year:

2010

Language:

english

File:

PDF, 426 KB

english, 2010

38

Constitutive activation of chimeric m2/m5 muscarinic receptors and delineation of G-protein coupling selectivity domains

Ethan S. Burstein, Tracy A. Spalding, Mark R. Brann

Journal:

Biochemical Pharmacology

Year:

1996

Language:

english

File:

PDF, 652 KB

english, 1996

39

Constitutively active muscarinic receptors

Tracy A. Spalding, Ethan S. Burstein

Journal:

Year:

2001

Language:

english

File:

PDF, 269 KB

english, 2001

40

Pharmacology of polymorphic variants of the human 5-HT1A receptor

Andria L. Del Tredici, Hans H. Schiffer, Ethan S. Burstein, Jelveh Lameh, Nina Mohell, Uli Hacksell, Mark R. Brann, David M. Weiner

Journal:

Biochemical Pharmacology

Year:

2004

Language:

english

File:

PDF, 270 KB

english, 2004

41

Studies of the Pharmacology, Localization, and Structure of Muscarinic Acetylcholine Receptors

MARK R. BRANN, HANS B. JØRGENSEN, ETHAN S. BURSTEIN, TRACY A. SPALDING, JOHN ELLIS, S. V. PENELOPE JONES, DAVID HILL-EUBANKS

Journal:

Annals of the New York Academy of Sciences

Year:

1993

Language:

english

File:

PDF, 659 KB

english, 1993

42

Estrogen Receptor Beta Selective Agonists as Agents to Treat Chemotherapeutic-Induced Neuropathic Pain

Ma, Jian-Nong, McFarland, Krista, Olsson, Roger, Burstein, Ethan S.

Journal:

ACS Chemical Neuroscience

Year:

2016

Language:

english

File:

PDF, 1.46 MB

english, 2016

43

Should inverse agonists be defined by pharmacological mechanism or clinical effect?

Burstein, Ethan S.

Journal:

Year:

2019

Language:

english

File:

PDF, 104 KB

english, 2019

44

I. In vivo evidence for partial agonist effects of (−)-OSU6162 and (+)-OSU6162 on 5-HT2A serotonin receptors

Maria L. Carlsson, Ethan S. Burstein, Angélica Kloberg, Sarah Hansson, Arja Schedwin, Marie Nilsson, Johan P. Rung, Arvid Carlsson

Journal:

Journal of Neural Transmission

Year:

2011

Language:

english

File:

PDF, 1.86 MB

english, 2011

45

The A-CD analogue of 16β,17α-estriol is a potent and highly selective estrogen receptor β agonist

Sauvée, Claire, Schäfer, Anja, Sundén, Henrik, Ma, Jian-Nong, Gustavsson, Anna-Lena, Burstein, Ethan S., Olsson, Roger

Journal:

Year:

2013

Language:

english

File:

PDF, 384 KB

english, 2013

46

Discovery of non-peptidergic MrgX1 and MrgX2 receptor agonists and exploration of an initial SAR using solid-phase synthesis

Leila Malik, Nicholas M. Kelly, Jian-Nong Ma, Erika A. Currier, Ethan S. Burstein, Roger Olsson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 1.54 MB

english, 2009

47

G-protein-coupled receptor-mediated activation of rap GTPases: characterization of a novel Gαi regulated pathway

Weissman, Jacques T, Ma, Jian-Nong, Essex, Anthony, Gao, Yan, Burstein, Ethan S

Journal:

Year:

2004

Language:

english

File:

PDF, 333 KB

english, 2004

48

Triazolam Kinetics: Interaction with Cimetidine, Propranolol, and the Combination

Friedman, H., Greenblatt, David J., Burstein, Ethan S., Scavone, Joseph M., Harmatz, Jerold S., Shader, Richard I.

Journal:

Journal of Clinical Pharmacology

Year:

1988

Language:

english

File:

PDF, 841 KB

english, 1988

49

The Second Intracellular Loop of the m5 Muscarinic Receptor Is the Switch Which Enables G-protein Coupling

Burstein, Ethan S., Spalding, Tracy A., Brann, Mark R.

Journal:

Journal of Biological Chemistry

Year:

1998

Language:

english

File:

PDF, 236 KB

english, 1998

50

AC-260584, an orally bioavailable M1 muscarinic receptor allosteric agonist, improves cognitive performance in an animal model

Stefania Risso Bradley, Jelveh Lameh, Linda Ohrmund, Thomas Son, Abhishek Bajpai, Derek Nguyen, Mikael Friberg, Ethan S. Burstein, Tracy A. Spalding, Thomas R. Ott, Hans H. Schiffer, Ali Tabatabaei, K

Journal:

Neuropharmacology

Year:

2010

Language:

english

File:

PDF, 910 KB

english, 2010

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